Dimerization of the Peptide CXCR4-Antagonist on Macromolecular and Supramolecular Protraction Arms Affords Increased Potency and Enhanced Plasma Stability. / Harms, Mirja; Hansson, Rikke Fabech; Carmali, Sheiliza; Almeida-Hernández, Yasser; Sanchez-Garcia, Elsa; Münch, Jan; Zelikin, Alexander N.
In: Bioconjugate Chemistry, Vol. 33, No. 4, 04.2022, p. 594-607.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Per-glycosylation of the Surface-Accessible Lysines : One-Pot Aqueous Route to Stabilized Proteins with Native Activity. / Walther, Raoul; Monge, Pere; Pedersen, Andreas; Benderoth, Anja; Pedersen, Jannik; Farzadfard, Azad; Mandrup, Ole; Howard, Kenneth; Otzen, Daniel; Zelikin, Alexander N.
In: ChemBioChem, Vol. 22, No. 14, 07.2021, p. 2478-2485.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Synthetic Artificial Apoptosis-Inducing Receptor for On-Demand Deactivation of Engineered Cells. / Monge, Pere; Løvschall, Kaja Borup; Søgaard, Ane Bretschneider; Walther, Raoul; Golbek, Thaddeus W.; Schmüser, Lars; Weidner, Tobias; Zelikin, Alexander N.
In: Advanced Science, Vol. 8, No. 13, 2004432, 07.2021.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Ceria Nanozyme and Phosphate Prodrugs : Drug Synthesis through Enzyme Mimicry. / Walther, Raoul; Huynh, Tin H.; Monge, Pere; Fruergaard, Anne Sofie; Mamakhel, Aref; Zelikin, Alexander N.
In: ACS Applied Materials and Interfaces, Vol. 13, No. 22, 06.2021, p. 25685-25693.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Antimicrobial activity of cyclic-monomeric and dimeric derivatives of the snail-derived peptide cm-p5 against viral and multidrug-resistant bacterial strains. / González-García, Melaine; Morales-Vicente, Fidel; Pico, Erbio Díaz; Garay, Hilda; Rivera, Daniel G.; Grieshober, Mark; Olari, Lia Raluca; Groß, Rüdiger; Conzelmann, Carina; Krüger, Franziska; Zech, Fabian; Bozzo, Caterina Prelli; Müller, Janis A.; Zelikin, Alexander; Raber, Heinz; Kubiczek, Dennis; Rosenau, Frank; Münch, Jan; Stenger, Steffen; Spellerberg, Barbara; Franco, Octavio L.; Alfonso, Armando A.Rodriguez; Ständker, Ludger; Otero-Gonzalez, Anselmo J.
In: Biomolecules, Vol. 11, No. 5, 745, 05.2021.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Carrageenan-containing over-the-counter nasal and oral sprays inhibit SARS-CoV-2 infection of airway epithelial cultures. / Schutz, Desiree; Conzelmann, Carina; Fois, Giorgio; Groß, Rudiger; Weil, Tatjana; Wettstein, Lukas; Stenger, Steffen; Zelikin, Alexander; Hoffmann, Thomas K.; Frick, Manfred; Muller, Janis A.; Munch, Jan.
In: American Journal of Physiology - Lung Cellular and Molecular Physiology, Vol. 320, No. 5, 05.2021, p. L750-L756.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Chemical (neo)glycosylation of biological drugs. / Walther, Raoul; Zelikin, Alexander N.
In: Advanced Drug Delivery Reviews, Vol. 171, 04.2021, p. 62-76.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Nitric Oxide to Fight Viral Infections. / Lisi, Fabio; Zelikin, Alexander N.; Chandrawati, Rona.
In: Advanced Science, Vol. 8, No. 7, 2003895, 04.2021.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Broad-Spectrum Antiviral Agents Based on Multivalent Inhibitors of Viral Infectivity. / Zelikin, Alexander N.; Stellacci, Francesco.
In: Advanced Healthcare Materials, Vol. 10, No. 6, 2001433, 03.2021.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Synthetic chemical ligands and cognate antibodies for biorthogonal drug targeting and cell engineering. / Monge, Pere; Søgaard, Ane Bretschneider; Andersen, Dante Guldbrandsen; Chandrawati, Rona; Zelikin, Alexander N.
In: Advanced Drug Delivery Reviews, Vol. 170, 03.2021, p. 281-293.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Nanozymes and Glucuronides : Glucuronidase, Esterase, and/or Transferase Activity. / Walther, Raoul; van den Akker, Wouter; Fruergaard, Anne Sofie; Zelikin, Alexander N.
In: Small, Vol. 16, No. 44, 2004280, 11.2020.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Artificial Biology : Molecular Design and Cell Mimicry. / Zelikin, Alexander N.; Städler, Brigitte.
In: Small, Vol. 16, No. 27, 2003442, 07.2020.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Editorial › Research › peer-review
Enzyme Mimics for the Catalytic Generation of Nitric Oxide from Endogenous Prodrugs. / Yang, Tao; Zelikin, Alexander N.; Chandrawati, Rona.
In: Small, Vol. 16, No. 27, 1907635, 07.2020.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Remotely Triggered Liquefaction of Hydrogel Materials. / Pedersen, Søren L.; Huynh, Tin H.; Pöschko, Philipp; Fruergaard, Anne Sofie; Jarlstad Olesen, Morten T.; Chen, Yaqing; Birkedal, Henrik; Subbiahdoss, Guruprakash; Reimhult, Erik; Thøgersen, Jan; Zelikin, Alexander N.
In: ACS Nano, Vol. 14, No. 7, 07.2020, p. 9145-9155.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Zinc Oxide Particles Catalytically Generate Nitric Oxide from Endogenous and Exogenous Prodrugs. / Yang, Tao; Fruergaard, Anne Sofie; Winther, Anna K.; Zelikin, Alexander N.; Chandrawati, Rona.
In: Small, Vol. 16, No. 27, 1906744, 07.2020.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
S-nitrosothiol-terminated poly(vinyl alcohol) : Nitric oxide release and skin blood flow response. / Giglio, Leonardo P.; Picheth, Guilherme F.; Løvschall, Kaja Borup; Zelikin, Alexander N.; de Oliveira, Marcelo G.
In: Nitric Oxide - Biology and Chemistry, Vol. 98, 05.2020, p. 41-49.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Molecular, macromolecular, and supramolecular glucuronide prodrugs : Lead identified for anticancer prodrug monotherapy. / Olesen, Morten Tobias Jarlstad; Walther, Raoul; Poier, Pier Paolo; Dagnæs-Hansen, Niels Frederik; Zelikin, Alexander N.
In: Angewandte Chemie International Edition, Vol. 59, No. 19, 02.2020, p. 7390-7396.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Unique enzymatic repertoire reveals the tumour. / Zelikin, Alexander N.
In: Nature Chemistry, Vol. 12, 01.2020, p. 11-12.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Comment/debate/letter to the editor › Research › peer-review
Chemical Artificial Internalizing Receptors for Primary T Cells. / Monge, Pere; Tvilum, Anne; Søgaard, Ane Bretschneider; Løvschall, Kaja Borup; Jarlstad Olesen, Morten T.; Zelikin, Alexander N.
In: Advanced Science, Vol. 7, No. 18, 2001395, 2020.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Inhaled and systemic heparin as a repurposed direct antiviral drug for prevention and treatment of COVID-19. / Conzelmann, Carina; Müller, Janis A.; Perkhofer, Lukas; Sparrer, Konstantin M.J.; Zelikin, Alexander N.; Münch, Jan; Kleger, Alexander.
In: Clinical Medicine, Vol. 20, No. 6, 2020, p. e218-e221.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Potent Lymphatic Translocation and Spatial Control Over Innate Immune Activation by Polymer–Lipid Amphiphile Conjugates of Small-Molecule TLR7/8 Agonists. / De Vrieze, Jana; Louage, Benoit; Deswarte, Kim; Zhong, Zifu; De Coen, Ruben; Van Herck, Simon; Nuhn, Lutz; Kaas Frich, Camilla; Zelikin, Alexander N.; Lienenklaus, Stefan; Sanders, Niek N.; Lambrecht, Bart N.; David, Sunil A.; De Geest, Bruno G.
In: Angewandte Chemie - International Edition, Vol. 58, No. 43, 10.2019, p. 15390-15395.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Delivering antibiotics locally to biofilms by targeted drug delivery and prodrug therapy. / Meyer, Rikke Louise; Walther, Raoul; Nielsen, Signe Maria; Andersen, Pernille Ommen; Hansen, Line; Vu-Quang, Hieu; Kjems, Jørgen; Zelikin, Alexander N.
2019. Abstract from Eurobiofilms 2019, Glasgow, United Kingdom.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
Extended scaffold glucuronides : en route to the universal synthesis of O-aryl glucuronide prodrugs. / Walther, Raoul; Olesen, Morten T. Jarlstad; Zelikin, Alexander N.
In: Organic & Biomolecular Chemistry, Vol. 17, No. 29, 08.2019, p. 6970-6974.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Non-covalent hitchhiking on endogenous carriers as a protraction mechanism for antiviral macromolecular prodrugs. / Frich, Camilla Kaas; Krüger, Franziska; Walther, Raoul; Domar, Cecilie; Andersen, Anna H. F.; Tvilum, Anne ; Dagnæs-Hansen, Frederik; Denton, Paul W.; Tolstrup, Martin; Paludan, Søren Riis; Münch, jJan; Zelikin, Alexander N.
In: Journal of Controlled Release, Vol. 294, 28.01.2019, p. 298-310.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Identification and Directed Development of Non‐Organic Catalysts with Apparent Pan‐Enzymatic Mimicry into Nanozymes for Efficient Prodrug Conversion. / Walther, Raoul; Winther, Anna; Fruergaard, Anne Sofie; Akker, Wouter van den; Sørensen, Lise; Nielsen, Signe Maria; Olesen, Morten Tobias Jarlstad; Dai, Yitao; Jeppesen, Henrik Særkjær; Lamagni, Paolo; Savateev, Aleksandra; Pedersen, Søren L.; Frich, Camilla Kaas; Vigier, Cécile Aude; Lock, Nina; Singh, Mandeep; Bansal, Vipul; Meyer, Rikke Louise; Zelikin, Alexander N.
In: Angewandte Chemie International Edition, Vol. 58, No. 1, 02.01.2019, p. 278-282.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Innate glycosidic activity in metallic implants for localized synthesis of antibacterial drugs. / Meer, Marja Ter; Dillion, Ross; Nielsen, Signe Maria; Walther, Raoul; Meyer, Rikke L.; Daamen, Willeke F.; Van Den Heuvel, Lambertus P.; Van Der Vliet, J. Adam; Lomme, Roger M.L.M.; Hoogeveen, Yvonne L.; Schultze Kool, Leo J.; Schaffer, Jeremy E.; Zelikin, Alexander N.
In: Chemical Communications, Vol. 55, No. 4, 01.01.2019, p. 443-446.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Antifouling properties of layer by layer DNA coatings. / Subbiahdoss, Guruprakash; Zeng, Guanghong; Aslan, Hüsnü; Ege Friis, Jakob; Iruthayaraj, Joseph; Zelikin, Alexander N.; Meyer, Rikke Louise.
In: Biofouling, Vol. 35, No. 1, 01.2019, p. 75-88.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Nucleic Acids as a Nature-Inspired Scaffold for Macromolecular Prodrugs of Nucleoside Analogues. / Krüger, Franziska; Kumar, Vipin; Monge, Pere; Conzelmann, Carina; Smith, Nikaïa; Gothelf, Kurt V.; Tolstrup, Martin; Münch, Jan; Zelikin, Alexander N.
In: Advanced Science, Vol. 6, No. 6, 1802095, 2019.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Combatting implant-associated biofilms through localized drug synthesis. / Walther, Raoul; Nielsen, Signe Maria; Christiansen, Rikke; Meyer, Rikke L.; Zelikin, Alexander N.
In: Journal of Controlled Release, Vol. 287, 10.10.2018, p. 94-102.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Development of an iron oxide nanoparticle drug delivery system against Staphylococcus aureus biofilm infections. / Dreier, Cindy; Zelikin, Alexander N.; Kjems, Jørgen; Meyer, Rikke Louise.
2018. Abstract from ICONAN2018, Rom, Italy.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
Bi‐Enzymatic Embolization Beads for Two‐Armed Enzyme‐Prodrug Therapy. / Olesen, Morten Tobias Jarlstad; Winther, Anna; Fejerskov, Betina; Dagnæs-Hansen, Frederik; Simonsen, Ulf; Zelikin, Alexander N.
In: Advanced Therapeutics, Vol. 1, No. 4, 1800023, 05.06.2018.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Progress and Promise of Nitric Oxide-Releasing Platforms. / Yang, Tao; Zelikin, Alexander N.; Chandrawati, Rona.
In: Advanced Science, Vol. 5, No. 6, 1701043, 01.06.2018.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Long-Acting, Potent Delivery of Combination Antiretroviral Therapy. / Andersen, Anna H. F.; Frich, Camilla Kaas; Zuwala, Kaja; Tolstrup, Martin; Dagnæs-Hansen, Frederik; Denton, Paul W.; Zelikin, Alexander N.
In: ACS Macro Letters, Vol. 7, No. 5, 30.04.2018, p. 587–591.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Letter › Research › peer-review
Enzyme Prodrug Therapy Achieves Site-Specific, Personalized Physiological Responses to the Locally Produced Nitric Oxide. / Winther, Anna K.; Fejerskov, Betina; Ter Meer, Marja; Jensen, Najah B.S.; Dillion, Ross; Schaffer, Jeremy E.; Chandrawati, Rona; Stevens, Molly M.; Schultze Kool, Leo J.; Simonsen, Ulf; Zelikin, Alexander N.
In: A C S Applied Materials and Interfaces, Vol. 10, No. 13, 04.04.2018, p. 10741-10751.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
The molecular tweezer CLR01 inhibits Ebola and Zika virus infection. / Röcker, Annika E.; Müller, Janis A.; Dietzel, Erik; Harms, Mirja; Krüger, Franziska; Heid, Christian ; Sowislok, Andrea ; Riber, Camilla Frich; Kupke, Alexandra; Lippold, Sina; von Einem, Jens; Beer, Judith; Knöll, Bernd; Becker, Stephan; Schmidt-Charnasit, Jonas; Otto, Markus; Vapalahti, Olli; Zelikin, Alexander N.; Bitan, Gal; Schrader, Thomas; Münch, Jan.
In: Antiviral Research, Vol. 152, 01.04.2018, p. 26-35.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Langstidsvirkende lægemidler via polymer-albumin-konjugation. / Frich, Camilla Kaas; Andersen, Anna H. F.; Zelikin, Alexander N.
In: Dansk Kemi, Vol. 99, No. 4, 2018, p. 10-12.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular prodrugs of ribavirin : Polymer backbone defines blood safety, drug release, and efficacy of anti-inflammatory effects. / Riber, Camilla Frich; Zuwala, Kaja; Løvschall, Kaja; Andersen, Anna H. F.; Sørensen, Lise; Gajda, Paulina; Tolstrup, Martin; Zelikin, Alexander N.
In: Journal of Controlled Release, Vol. 275, No. April, 2018, p. 53-66.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular Antiviral Agents against Zika, Ebola, SARS, and Other Pathogenic Viruses. / Schandock, Franziska; Riber, Camilla Frich; Röcker, Annika; Müller, Janis A; Harms, Mirja; Gajda, Paulina; Zuwala, Kaja; Andersen, Anna H F; Løvschall, Kaja Borup; Tolstrup, Martin; Kreppel, Florian; Münch, Jan; Zelikin, Alexander N.
In: Advanced Healthcare Materials, 12.2017.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Enzyme Prodrug Therapy Engineered into Electrospun Fibers with Embedded Liposomes for Controlled, Localized Synthesis of Therapeutics. / Chandrawati, Rona; Olesen, Morten T. J.; Marini, Thatiane C. C.; Bisra, Gurpal; Guex, Anne Geraldine; de Oliveira, Marcelo G.; Zelikin, Alexander N.; Stevens, Molly M.
In: Advanced Healthcare Materials, Vol. 6, No. 17, 1700385, 06.09.2017.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Enzyme prodrug therapies and therapeutic enzymes. / Städler, Brigitte; Zelikin, Alexander N.
In: Advanced Drug Delivery Reviews, Vol. 118, No. 9, 01.09.2017.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Editorial › Research › peer-review
Prodrugs in medicinal chemistry and enzyme prodrug therapies. / Walther, Raoul; Rautio, Jarkko; Zelikin, Alexander N.
In: Advanced Drug Delivery Reviews, Vol. 118, No. september, 01.09.2017, p. 65-77.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Synthetic Polymer with a Structure-Driven Hepatic Deposition and Curative Pharmacological Activity in Hepatic Cells. / Riber, Camilla Frich; Halling Folkmar Andersen, Anna; Anegaard Rolskov, Lærke ; Zuwala, Kaja; Gajda, Paulina; Borup Løvschall, Kaja; Dagnæs-Hansen, Frederik; Banda, Dominic H.; Pietschmann, Thomas; Tolstrup, Martin; Zelikin, Alexander N.
In: ACS Macro Letters, Vol. 6, No. 935-940, 15.08.2017, p. 935-940.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Preparation, single-molecule manipulation and energy transfer investigation of a polyfluorene-graft-DNA polymer. / Madsen, Mikael; Christensen , Rasmus S. ; Krissanaprasit, Abhichart; Bakke, Mette Riis; Riber, Camilla Frich; Nielsen , Karina S. ; Zelikin, Alexander N.; Gothelf, Kurt Vesterager.
In: Chemistry: A European Journal, Vol. 23, No. 44, 22.06.2017.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Recent advances in macromolecular prodrugs. / Riber, Camilla Frich; Zelikin, Alexander N.
In: Current Opinion in Colloid & Interface Science, Vol. 31, 21.06.2017.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Localized and Controlled Delivery of Nitric Oxide to the Conventional Outflow Pathway via Enzyme Biocatalysis : Toward Therapy for Glaucoma. / Chandrawati, Rona; Chang, Jason Y. H.; Reina-Torres, Ester; Jumeaux, Coline; Sherwood, Joseph M.; Stamer, W. Daniel; Zelikin, Alexander N.; Overby, Darryl R.; Stevens, Molly M.
In: Advanced Materials, Vol. 29, No. 16, 1604932, 25.04.2017.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular Prodrugs of Ribavirin : Structure-Function Correlation as Inhibitors of Influenza Infectivity. / Riber, Camilla Frich; Hinton, Tracey M; Gajda, Paulina; Zuwala, Kaja; Tolstrup, Martin; Stewart, Cameron; Zelikin, Alexander N.
In: Molecular Pharmaceutics, Vol. 14, No. 1, 03.01.2017, p. 234-241.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Substrate mediated enzyme prodrug therapy. / Fejerskov, Betina; Jarlstad Olesen, Morten T; Zelikin, Alexander N.
In: Advanced Drug Delivery Reviews, Vol. 118, 2017, p. 24-34.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research › peer-review
Albumin–Polymer–Drug Conjugates: Long Circulating, High Payload Drug Delivery Vehicles. / Smith, Anton Allen Abbotsford; Zuwala, Kaja; Pilgram, Oliver; Johansen, Karen Singers Eiskjær; Tolstrup, Martin; Dagnæs-Hansen, Frederik; Zelikin, Alexander N.
In: ACS Macro Letters, Vol. 5, 15.09.2016, p. 1089-1094.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Poly(vinyl alcohol) Physical Hydrogels : Matrix-Mediated Drug Delivery Using Spontaneously Eroding Substrate. / Jensen, Bettina E. B.; Davila, Izaskun; Zelikin, Alexander N.
In: Journal of Physical Chemistry Part B: Condensed Matter, Materials, Surfaces, Interfaces & Biophysical, Vol. 120, No. 26, 07.07.2016, p. 5916-5926.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Triple Activity of Lamivudine Releasing Sulfonated Polymers against HIV-1. / Danial, Maarten; Halling Folkmar Andersen, Anna; Zuwala, Kaja; Cosson, Steffen; Riber, Camilla Frith; Smith, Anton A. A.; Tolstrup, Martin; Moad, Graeme; Zelikin, Alexander N.; Postma, Almar.
In: Molecular Pharmaceutics, Vol. 13, No. 7, 07.2016, p. 2397-2410.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
HIV anti-latency treatment mediated by macromolecular prodrugs of histone deacetylase inhibitor, panobinostat. / Zuwala, Kaja; Smith, Anton Allen Abbotsford; Tolstrup, Martin; Zelikin, Alexander N.
In: Chemical Science, Vol. 7, No. 3, 2016, p. 2353-2358.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Materials and methods for delivery of biological drugs. / Zelikin, Alexander N.; Ehrhardt, Carsten; Healy, Anne Marie.
In: Nature Chemistry, Vol. 8, No. 11, 2016, p. 997-1007.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Polyanionic Macromolecular Prodrugs of Ribavirin : Antiviral Agents with a Broad Spectrum of Activity. / Hinton, Tracey M.; Zuwala, Kaja; Deffrasnes, Celine; Todd, Shawn; Shi, Shuning; Marsh, Glenn A.; Dearnley, Megan; Wohl, Benjamin M.; Tolstrup, Martin; Zelikin, Alexander N.
In: Advanced Healthcare Materials, Vol. 5, No. 5, 2016, p. 534-540.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Tools of gene transfer applied to the intracellular delivery of non-nucleic acid polyanionic drugs. / Kryger, Mille B. L.; Pedersen, Søren L.; Wohl, Benjamin M.; Zelikin, Alexander N.
In: Chemical Communications, Vol. 52, No. 5, 2016, p. 889-891.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Routing of individual polymers in designed patterns. / Knudsen, Jakob Bach; Liu, Lei; Kodal, Anne Louise Bank; Madsen, Mikael; Li, Qiang; Song, Jie; Woehrstein, Johannes; Wickham, Shelley; Strauss, Maximillian; Schueder, Florian; Vinther, Jesper; Krissanaprasit, Abhichart; Gudnason, Daniel Aron; Smith, Anton Allen Abbotsford; Ogaki, Ryosuke; Zelikin, Alexander N.; Besenbacher, Flemming; Birkedal, Victoria; Yin, Peng; Shih, William M.; Jungmann, Ralf; Dong, Mingdong; Gothelf, Kurt Vesterager.
In: Nature Nanotechnology, Vol. 10, 31.08.2015, p. 892-898.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Self-Immolative Linkers Literally Bridge Disulfide Chemistry and the Realm of Thiol-Free Drugs. / Riber, Camilla Frich; Smith, Anton A. A.; Zelikin, Alexander N.
In: Advanced Healthcare Materials, Vol. 4, No. 12, 26.08.2015, p. 1887-1890.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Micro-structured, spontaneously eroding hydrogels accelerate endothelialization through presentation of conjugated growth factors. / Jensen, Bettina E. B.; Edlund, Katrine; Zelikin, Alexander N.
In: Biomaterials, Vol. 49, 05.2015, p. 113-124.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Highly active macromolecular prodrugs inhibit expression of the hepatitis c virus genome in the host cells. / Ruiz-Sanchis, Pau; Wohl, Benjamin M.; Smith, Anton A A; Zuwala, Kaja; Melchjorsen, Jesper; Tolstrup, Martin; Zelikin, Alexander N.
In: Advanced Healthcare Materials, Vol. 4, No. 1, 01.01.2015, p. 65-68.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular prodrugs of ribavirin : towards a treatment for co-infection with HIV and HCV. / Smith, Anton Allen Abbotsford; Zuwala, Kaja; Kryger, Mille; Wohl, Benjamin; Guerrero-Sanchez, Carlos; Tolstrup, Martin; Postma, Almar; Zelikin, Alexander N.
In: Chemical Science, Vol. 6, No. 1, 2015, p. 264-269.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Phospholipid-polymer amphiphile hybrid assemblies and their interaction with macrophages. / Panneerselvam, Karthiga; Lynge, Martin E.; Riber, Camilla Frich; Mena-Hernando, Sofia; Smith, Anton A. A.; Goldie, Kenneth N.; Zelikin, Alexander N.; Stadler, Brigitte.
In: Biomicrofluidics, Vol. 9, No. 5, 052610, 2015.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Polymers Fight HIV : Potent (Pro)Drugs Identified Through Parallel Automated Synthesis. / Zuwala, Kaja; Smith, Anton A A; Postma, Almar; Guerrero-Sanchez, Carlos; Ruiz Sanchis, Pau; Melchjorsen, Jesper; Tolstrup, Martin; Zelikin, Alexander N.
In: Advanced Healthcare Materials, Vol. 4, No. 1, 2015, p. 46-50.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Disulfide reshuffling triggers the release of a thiol-free anti-HIV agent to make up fast-acting, potent macromolecular prodrugs. / Kock, Anders; Zuwala, Kaja; Smith, Anton A A; Ruiz-Sanchis, Pau; Wohl, Benjamin M; Tolstrup, Martin; Zelikin, Alexander N.
In: Chemical Communications, Vol. 50, No. 93, 04.12.2014, p. 14498-500.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Enzyme prodrug therapy engineered into biomaterials. / Mendes, Ana C.; Zelikin, Alexander N.
In: Advanced Functional Materials, Vol. 24, No. 33, 03.09.2014, p. 5202-5210.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Biocatalytic polymer thin films : optimization of the multilayered architecture towards in situ synthesis of anti-proliferative drugs. / Andreasen, Sidsel Ø; Fejerskov, Betina; Zelikin, Alexander N.
In: Nanoscale, Vol. 6, No. 8, 21.04.2014, p. 4131-40.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Biocatalytic polymer coatings : on-demand drug synthesis and localized therapeutic effect under dynamic cell culture conditions. / Fejerskov, Betina; Jensen, Najah B S; Mian Teo, Boon; Stadler, Brigitte Maria; Zelikin, Alexander N.
In: Small, Vol. 10, No. 7, 09.04.2014, p. 1314-24.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular Prodrugs of Ribavirin: Concerted Efforts of the Carrier and the Drug. / Smith, Anton A A; Wohl, Benjamin M; Kryger, Mille B L; Hedemann, Natasha; Guerrero-Sanchez, Carlos; Postma, Almar; Zelikin, Alexander N.
In: Advanced Healthcare Materials, Vol. 3, No. 9, 10.01.2014, p. 1404-1407.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular (pro)Drugs in antiviral research. / Smith, Anton Allen Abbotsford; Kryger, Mille; Wohl, Benjamin; Ruiz Sanchis, Pau; Zuwala, Kaja; Tolstrup, Martin; Zelikin, Alexander N.
In: Polymer Chemistry, Vol. 5, No. 22, 2014, p. 6407-6425.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular (pro)drugs with concurrent direct activity against the hepatitis C virus and inflammation. / Wohl, Benjamin; Smith, Anton Allen Abbotsford; Jensen, Bettina Elisabeth Brøgger; Zelikin, Alexander N.
In: Journal of Controlled Release, Vol. 196, 2014, p. 197–207.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular Prodrugs for Controlled Delivery of Ribavirin. / Kryger, Mille B L; Smith, Anton A A; Wohl, Benjamin M; Zelikin, Alexander N.
In: Macromolecular Bioscience, Vol. 14, No. 2, 2014, p. 173-185.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Cholesterol Modification of (Bio)Polymers Using UV-Vis Traceable Chemistry in Aqueous Solutions. / Rasmussen, Kasper F; Smith, Anton A A; Ruiz-Sanchis, Pau; Edlund, Katrine; Zelikin, Alexander N.
In: Macromolecular Bioscience, Vol. 14, No. 1, 17.09.2013, p. 33-44.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Poly(vinyl alcohol) Physical Hydrogel Nanoparticles, Not Polymer Solutions, Exert Inhibition of Nitric Oxide Synthesis in Cultured Macrophages. / Andreasen, Sidsel Østerby; Chong, Siow Feng; Wohl, Benjamin M; Goldie, Kenneth N; Zelikin, Alexander N.
In: Biomacromolecules, Vol. 14, 22.04.2013, p. 1687-1695.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecular prodrugs of ribavirin combat side effects and toxicity with no loss of activity of the drug. / Kryger, M.B.L.; Wohl, B.M.; Smith, A.A.A.; Zelikin, Alexander N.
In: Chemical Communications, Vol. 49, No. 26, 04.04.2013, p. 2643-2645.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Bioresorbable Surface-Adhered Enzymatic Microreactors Based on Physical Hydrogels of Poly(vinyl alcohol). / Fejerskov, Betina; Smith, Anton A A; Jensen, Bettina E B; Hussmann, Thomas; Zelikin, Alexander N.
In: Langmuir, Vol. 29, No. 1, 2013, p. 344-54.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Lipogels: Surface-Adherent Composite Hydrogels Assembled from Poly(Vinyl Alcohol) and Liposomes. / Jensen, Bettina Elisabeth Brøgger; Rigau, Leticia Hosta; Spycher, Philipp; Reimhult, Erik; Stadler, Brigitte Maria; Zelikin, Alexander N.
In: Nanoscale, Vol. 5, No. 15, 2013, p. 6758-6766.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Liposomal Templating, Association with Mammalian Cells, and Cytotoxicity of Poly(vinyl alcohol) Physical Hydrogel Nanoparticles. / Andreasen, Sidsel Østerby; Chong, Siow Feng; Kryger, Mille; Jensen, Bettina Elisabeth Brøgger; Postma, Almar; Alves, Marie-Helene; Stadler, Brigitte Maria; Goldie, Kenneth; Zelikin, Alexander N.
In: Particle & Particle Systems Characterization, Vol. 30, No. 6, 2013, p. 514-522.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Liposomes as Drug Deposits in Multilayered Polymer Films. / Madsen, Martin Elias Lynge; Laursen, Marie Bækgaard; Rigau, Leticia Hosta; Jensen, Bettina Elisabeth Brøgger; Ogaki, Ryosuke; Smith, Anton Allen Abbotsford; Zelikin, Alexander N.; Stadler, Brigitte Maria.
In: A C S Applied Materials and Interfaces, Vol. 5, No. 8, 2013, p. 2967-2975.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Microstructured, Functional PVA Hydrogels through Bioconjugation with Oligopeptides under Physiological Conditions. / Chong, Siow Feng; Smith, Anton A A; Zelikin, Alexander N.
In: Small, Vol. 9, No. 6, 2013, p. 942-950.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Narrow Therapeutic Window of Ribavirin as an Inhibitor of Nitric Oxide Synthesis is Broadened by Macromolecular Prodrugs. / Wohl, Benjamin M; Smith, Anton Allen Abbotsford; Kryger, Mille B L; Zelikin, Alexander N.
In: Biomacromolecules, Vol. 14, No. 11, 2013, p. 3916-26.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Surface Grafted Glycopolymer Brushes to Enhance Selective Adhesion of HepG2 Cells. / Chernyy, Sergey; Jensen, Bettina Elisabeth Brøgger; Shimizu, Kyoko; Ceccato, Marcel; Pedersen, Steen Uttrup; Zelikin, Alexander N.; Daasbjerg, Kim; Iruthayaraj, Joseph.
In: Journal of Colloid and Interface Science, Vol. 404, 2013, p. 207–214.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Intelligent Polymer Thin Films and Coatings for Drug Delivery. / Zelikin, Alexander N.; Stadler, Brigitte Maria.
Intelligent Surfaces in Biotechnology - Scientific and engineering concepts, enabling technologies, and translation to bio-oriented applications. ed. / H. Michelle Grandin; Marcus Textor. John Wiley & Sons Ltd, 2012.Research output: Contribution to book/anthology/report/proceeding › Book chapter › Research › peer-review
Macromolecular design of poly(vinyl alcohol) by RAFT polymerization. / Smith, A.A.A.; Hussmann, Thomas; Elich, Joseph; Alves, Marie-Helene; Postma, A.; Zelikin, Alexander N.
In: Polymer Chemistry, Vol. 3, No. 1, 01.01.2012, p. 85-88.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Biodistribution of polymer hydrogel capsules for the delivery of therapeutics. / Hinton, Tracey M; Monaghan, Paul; Green, Diane; Kooijmans, Sander A A; Shi, Shuning; Breheney, Kerry; Tizard, Mark; Nicolazzo, Joseph A; Zelikin, Alexander N.; Wark, Kim.
In: Acta Biomaterialia, Vol. 8, No. 9, 2012, p. 3251-60.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Engineering surface adhered poly(vinyl alcohol) physical hydrogels as enzymatic microreactors. / Fejerskov, Betina; Jensen, Bettina E B; Jensen, Najah Brok Søndervang; Chong, Siow Feng; Zelikin, Alexander N.
In: A C S Applied Materials and Interfaces, Vol. 4, No. 9, 2012, p. 4981-90.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Macromolecule Functionalization of Disulfide-Bonded Polymer Hydrogel Capsules and Cancer Cell Targeting. / Shimoni, Olga; Postma, Almar; Yan, Yan; Scott, Andrew M.; Heath, Joan K.; Nice, Edouard C.; Zelikin, Alexander N.; Caruso, Frank.
In: A C S Nano, Vol. 6, No. 2, 2012, p. 1463-1472.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Substrate mediated enzyme prodrug therapy. / Fejerskov, Betina; Zelikin, Alexander N.
In: P L o S One, Vol. 7, No. 11, 2012, p. e49619.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Surface adhered poly(vinyl alcohol) physical hydrogels as tools for rational design of intelligent biointerfaces. / Jensen, Bettina Elisabeth Brøgger; Alves, Marie-Helene ; Fejerskov, Betina; Stadler, Brigitte; Zelikin, Alexander N.
In: Soft Matter, Vol. 8, 2012, p. 4625-4634.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Surface-Adhered Composite Poly(Vinyl Alcohol) Physical Hydrogels: Polymersome-Aided Delivery of Therapeutic Small Molecules. / Rigau, Leticia Hosta; Jensen, Bettina Elisabeth Brøgger; Fjeldsø, Kit; Postma, Almar; Li; Goldie; Albericio, ; Zelikin, Alexander N.; Stadler, Brigitte Maria.
In: Advanced Healthcare Materials, 2012.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
A Critical Look at multilayered Polymer Capsules in Biomedicine: Drug Carriers, Artificial organelles, and Cell Mimic. / Stadler, Brigitte; Price, Andrew D.; Zelikin, Alexander N.
In: Advanced Functional Materials, Vol. 21, No. 1, 07.01.2011, p. 14-28.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Degradation of liposomal subcompartments in PEGylated capsosomes. / Chandrawati, R.; Chong, S.-F.; Zelikin, Alexander N.; Rigau, Leticia Hosta; Stadler, Brigitte; Caruso, F.
In: Soft Matter, Vol. 8, 2011, p. 9638-9646.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Exploiting Fluorescent Polymers To Probe the Self-Assembly of Virus-like Particles. / Caden-Nava, Ruben D.; Hu, Yufang; Garmann, Rees F.; Ng, Benny; Zelikin, Alexander N.; Knobler, Charles M.; Gelbart, William M.
In: Journal of Physical Chemistry Part B: Condensed Matter, Materials, Surfaces, Interfaces & Biophysical, Vol. 115, 2011, p. 2386-2391.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Poly(vinyl alcohol) Physical Hydrogels: Non-cryogenic Stabilization Allows Nano- and Micro-Scale Materials Design. / Jensen, Bettina Elisabeth Brøgger; Smith, Anton Allen Abbotsford; Fejerskov, Betina; Postma, Almar; Senn, Philipp; Reimhult, Erik; Pla-Roca, Mateu; Isa, Lucio; Sutherland, Duncan S; Stadler, Brigitte; Zelikin, Alexander N.
In: Langmuir, Vol. 27, No. 16, 2011, p. 10216–10223.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Poly(vinyl alcohol) physical hydrogels : New vista on a long serving biomaterial. / Alves, M.-H.; Jensen, Bettina Elisabeth Brøgger; Smith, Anton Allen Abbotsford; Zelikin, Alexander N.
In: Macromolecular Bioscience, Vol. 11, 2011, p. 1293-1313.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Redox-Active Polymer Microcapsules for the Delivery of a Survivin-Specific siRNA in Prostate Cancer Cells. / Becker, A. L.; Orlotti, N. I. ; Folini, M.; Cavalieri, F.; Zelikin, Alexander N.; Johnston, A. P. R. J.; Zaffaroni, N.; Caruso, F.
In: ACS Nano, Vol. 5, 2011, p. 1335-1344.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Tuning the Permeability of Polymer Hydrogel Capsules: An Investigation of Cross-Linking Density, Membrane Thickness, and Cross-Linkers. / Chong, S.-F.; Zelikin, Alexander N.; Lee, J. H.; Caruso, F.
In: Langmuir, Vol. 27, 2011, p. 1724-1730.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Journal article › Research › peer-review
Drug Releasing Polymer Thin Films: New Era of Surface-Mediated Drug Delivery. / Zelikin, Alexander N.
In: A C S Nano, Vol. 4, No. 5, 2010, p. 2494-2509.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research
Poly(Methacrylic Acid) Polymer Hydrogel Capsules: Drug Carriers, Sub-compartmentalized Microreactors, Artificial Organelles. / Zelikin, Alexander N.; Price, Andrew; Stadler, Brigitte.
In: Small, Vol. 6, No. 20, 2010, p. 2201-2207.Research output: Contribution to journal/Conference contribution in journal/Contribution to newspaper › Review › Research