Keyphrases
Orthosteric Site
100%
Non-competitive Inhibitor
100%
Cryo-EM Structure
100%
Dopamine Transporter
100%
Dopamine
100%
Cocaine
100%
Transmembrane Domain
100%
Ectodomain Shedding
100%
Sortilin
100%
Domain-domain Interaction
100%
AC-4
66%
Amphetamine
66%
Psychostimulant Drugs
33%
Vestibule
33%
Non-competitive Inhibition
33%
Cryo-electron Microscopy Structure
33%
Rewarding Effect
33%
Attenuation
33%
Neurotransmitter Signaling
33%
Open Conformation
33%
Binding Site
33%
Sodium Chloride
33%
Synaptic Cleft
33%
Promising Strategies
33%
Drug Use Disorder
33%
Drosophila Melanogaster
33%
Rational Design
33%
Alzheimer's Disease
8%
Coarse-grained Molecular Dynamics Simulation
8%
Structural Framework
8%
Central Region
8%
Complex Formation
8%
Mutagenesis
8%
Neurotrophin Signaling
8%
Biochemical Assay
8%
Proteolysis
8%
Functional Specificity
8%
ADAM10
8%
Interaction Interface
8%
Molecular Control
8%
Structural Modeling
8%
Proteolytic Processing
8%
NSG2
8%
Metalloproteinases
8%
Disintegrin
8%
Selective Modulators
8%
Membrane Receptors
8%
Binding Mode
8%
Intracellular Trafficking
8%
Neuronal Proteins
8%
Biochemistry, Genetics and Molecular Biology
Dopamine Transporter
100%
Ectodomain
100%
Transmembrane Domain
100%
Cryoelectron Microscopy
100%
Competitive Inhibition
100%
Neurotransmitter
33%
Non-Competitive Inhibition
33%
Binding Site
33%
Drosophila Melanogaster
33%
ADAM10
16%
Proteolysis
16%
Complex Formation
16%
Proteolytic Processing
16%
Disintegrin
16%
Mutagenesis
16%
Metalloproteinase
16%
Intracellular Trafficking
16%
Transmembrane Receptors
16%
Metalloendopeptidase
16%
Neuroscience
Competitive Inhibition
100%
Cryo-Electron Microscopy
100%
Dopamine Transporter
100%
Amphetamine
66%
Vestibule of the Ear
33%
Psychostimulant
33%
Neurotransmitter
33%
Drosophila Melanogaster
33%
Binding Site
33%
Cleft
33%
Non-Competitive Inhibition
33%